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NALOXONE
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DeCS
Descriptor
English
:
Naloxone
Descriptor
Spanish
:
Naloxona
Descriptor
Portuguese
:
Naloxona
Tree Number:
D03.132.577.249.706
D03.549.686.750
D03.605.497.750
D04.615.723.795.706
Definition
English
:
A specific opiate antagonist that has no agonist activity. It is a competitive antagonist at mu,
delta
, and kappa opioid receptors.
Pharmacological Action:
Narcotic Antagonists
History Note
English
:
1973(1972); for MRZ-2593 use OXYMORPHONE 1985-2009
Allowable Qualifiers
English
:
AD
administration & dosage
AE
adverse effects
AG
agonists
AA
analogs & derivatives
AN
analysis
AI
antagonists & inhibitors
BL
blood
CF
cerebrospinal fluid
CS
chemical synthesis
CH
chemistry
CL
classification
CT
contraindications
DU
diagnostic use
EC
economics
HI
history
IM
immunology
IP
isolation & purification
ME
metabolism
PK
pharmacokinetics
PD
pharmacology
PO
poisoning
RE
radiation effects
ST
standards
SD
supply & distribution
TU
therapeutic use
TO
toxicity
UR
urine
Record Number:
9462
Unique Identifier:
D009270
Occurrence in VHL
:
Similar:
DeCS
CID-10
SciELO
LILACS
LIS